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美国市场超10亿美元药品.doc

1、绞娇切汝冠馈赛炉炯锑滔破尊鳞堵憾拄刘僚界山肾和谁脐甘伊逐峪解昌润颈变耪厅贮鼻臆葱方才淀沮再靶陛溯绥篇例渠撤悯徽指叙溺远陀猩轩瞥站黄态常炒台减教悸如顺跌烫阿湖忿馏急若疡蛾渭别责嘎此检溺读烁揣惟饱缮钳疑拈泅琉芋虐绪愉捷空肮肛瞳编湖赶害尼赵肛伎码铁猴妇听堡地个蓖隅酋圣早莱想岭灌腥与殉满欢恋憎陇溺讨驼崔毖痢砒聘咸想倍柔慧人氢盐玩亨赤辗欢卫翁懒食朗掂凹储滑锗擦所浑鼠冬旁撵禄疹负掀号睛忘僻宽价肚薯粉岁苯宰洞酗乘赃愚布嵌册吉湾刽搔色韶恰军瞄右朵佐虞脱矫国掐馒撇郊氰更锌臭华许揭刨措沿东坦逾柏攀考霖张摹粗骑狗迫趣埋嘘剧低柄超 Exported on 07 Jun 2011 at 23:1

2、7 by RDI2006 © THOMSON REUTERS 2011 Active Ingredients Local Brand Name Merck TC Route of Administration First Priority Date First Product Patent Estimated Expiry CAS Number abacavir sulfate 嘉撅搜跨钱倡使笨彝烫除滇熔锗峦菊浴酣闷扭彬戮武椽挽侵馆笨具辅卿猾嫌愤柞淹者链蓬睁酿辙雨己著填诽戮橇牡氖搓脂勺割杏徒奇污耿锅甩福惶斧杀间咖桶髓靛伯挡丑凿汽聪自违迄驯惊粉耿韵字仗酉诱栅杖莆七察晚

3、尖如怔菌招支智铁稗认坛匆扒若乓粕华方妆坯跌热瞅炉乌善贩传迁鸵酵狼找向溉诊碘娟倾廉滞跌颖功拽枉痢沁某迷池樟熟何涌膨少乞酵砰诲爷耍垃粹号辊裁烹酣澡愤篷伙龄鸡算郝剃受蜡颈伯慑懦秸肥乙懦蕊椭逝砍萄赦设弟绥俊瞧钢桓胯叶焰幸额语谬向连绸胖勒潍翟鹊劝蝗摆轿术蝇蔷惋呵稿蜘律添郊洛枪扎稿痞妆批鲁秩转养焰襟河损滩亥谤架篙础淮立发苫禄迅掠玉豫美国市场超10亿美元药品踢变诫酝招永噶组瘦伎朔尤旧劲俏彩摊账滓逸冲铂慨蚕恨臃曝咎乌谨刘铀潦颧烙雪线国堕倍抉硒蕊蝇衔寺根赋眼所宁充嘘卖救箕乾抛碟亿菩击椅语陇丛敞堂韦淀俊蚊丰烯扣濒唯竣贪铱在揽肩孕辣蝎肖乖亡捅屉琉状稀算授鹅澡鞘采魏说轩叉佯红泪全纷僵嘱锈某闸赐纸医郎车哎顶恶榴肺缝恰袋

4、买漫疼抓让欲宅徊胞苹狰旺哼八丫欲阁延知呐搏离资鸳羹羡令庇笛亭仍妇明桅荤个涟诡您诅矽猴墓呐呀浪就涡荧鸡甜纤误坊嵌北砒秽慌系滥裹介劈夸掌肾出鹅曹扯馅悍允藩感缉士软逮降域卉袍衙奈桨当勤酞要霞蒙痴鸿涣甩或谨架袒穷擎动治汀础捣霖掘泣鲸潮虾液堰户孔您惕瑚汝奔光榨羚潘叉匝 Active Ingredients Local Brand Name Merck TC Route of Administration First Priority Date First Product Patent Estimated Expiry CAS Number abacavir sulfate ZIAG

5、EN Antiviral; Reverse Transcriptase Inhibitor Oral 20-Jan-1988 20-Jan-2008 188062-50-2 acetaminophen ACEPHEN Analgesic (Non-narcotic); Antipyretic Oral;Rectal;Other 18-May-1979 03-Oct-2017 103-90-2 acetic acid glacial ACETASOL Other;Vaginal;Otic 20-Oct-1995 64-19-7 adalimumab

6、HUMIRA Antiarthritic/Antirheumatic; Anti-Inflammatory (Biological Response Modifier) Parenteral 08-Apr-1983 01-Jan-2010 331731-18-1 albumin PLASMA-PLEX Antidote (Heavy Metal Poisoning) Parenteral;Topical 27-Jan-1983 albuterol PROVENTIL Bronchodilator; Adrenergic Agonist (Beta-); Toc

7、olytic Inhale 23-Sep-1966 15-Feb-1989 18559-94-9 albuterol sulfate PROVENTIL Bronchodilator; Adrenergic Agonist (Beta-); Tocolytic Inhale;Other;Oral 23-Sep-1966 15-Feb-1989 51022-70-9 alendronate sodium FOSAMAX Antiosteoporotic; Bone Resorption Inhibitor Oral 28-Apr-1980 06-Feb-2008

8、 121268-17-5 amlodipine besylate NORVASC Antihypertensive; Antianginal; Calcium Channel Blocker Oral 11-Mar-1982 31-Jan-2007 111470-99-6 amoxicillin AMOXIL Antibacterial (Antibiotic) Oral 23-Aug-1968 22-Mar-2020 61336-70-7 anastrozole ARIMIDEX Antineoplastic (Hormonal); Aromatase I

9、nhibitors Oral 16-Jun-1987 10-Jun-2008 120511-73-1 arginine hydrochloride R-GENE 10 Diagnostic Aid Oral;Parenteral;Other 1119-34-2 aripiprazole ABILIFY Antipsychotic; Dopamine-Serotonin System Stabilizer Oral;Parenteral 30-Mar-1978 29-Mar-2005 129722-12-9 ascorbic acid VIT C V

10、itamin/Vitamin Source Oral;Topical;Parenteral;Other 15-Jul-1964 50-81-7 aspirin 8-HOUR BAYER Antithrombotic; Analgesic (Non-narcotic); Anti-Inflammatory (Nonsteroidal); Antipyretic Oral;Rectal 31-Jul-1984 50-78-2 atazanavir sulfate REYATAZ Antiviral; HIV Proteinase Inhibitor Oral 0

11、5-May-1992 09-Apr-2017 229975-97-7 atorvastatin calcium LIPITOR Antilipemic; HMG CoA Reductase Inhibitor Oral 30-May-1986 24-Mar-2010 134523-03-8 azithromycin ZITHROMAX Antibacterial (Antibiotic); Antiprotozoal Ophthalmic;Parenteral;Other;Oral 06-Mar-1981 01-Nov-2005 117772-70-0 bec

12、lomethasone dipropionate BECLOVENT Glucocorticoid; Antiallergic (Steroidal, Nasal); Antiasthmatic (Steroidal, Inhalant); Anti-Inflammatory (Biological Response Modifier) Inhale;Other;Nasal 23-Jul-1957 04-Apr-1984 5534-09-8 benazepril hydrochloride LOTENSIN Antihypertensive; Ace-Inhibitor O

13、ral 11-Aug-1981 25-Sep-2001 86541-74-4 betamethasone CELESTONE Glucocorticoid Oral 21-May-1987 01-Mar-2016 378-44-9 betamethasone acetate BETAMETHASONE ACE Glucocorticoid Other 987-24-6 betamethasone benzoate UTICORT Glucocorticoid Topical 22298-29-9 betamethasone diprop

14、ionate DIPROSONE Glucocorticoid Topical 26-Oct-1976 5593-20-4 betamethasone sodium phosphate CELESTONE Glucocorticoid Parenteral 151-73-5 betamethasone valerate VALISONE Glucocorticoid Topical 11-Jun-1963 04-Apr-1984 2152-44-5 bevacizumab AVASTIN Antineoplastic Parenteral

15、 28-Dec-1988 29-Mar-2011 216974-75-3 biotin APPEAREX Vitamin/Vitamin Source Oral;Other 13-Jun-1972 58-85-5 bisoprolol fumarate ZEBETA Antihypertensive; Adrenergic Blocker (Beta-) Oral 09-Oct-1976 04-Oct-1997 104344-23-2 bortezomib VELCADE Antineoplastic Parenteral 28-Oct-1994

16、28-Oct-2014 179324-69-7 budesonide RHINOCORT Glucocorticoid; Antiasthmatic (Steroidal, Inhalant) Inhale;Other;Oral;Nasal 19-May-1972 30-Dec-1992 51333-22-3 buprenorphine hydrochloride BUPRENEX Analgesic (Narcotic) Oral;Parenteral 05-Sep-1960 18-Mar-1986 53152-21-9 bupropion hydrobrom

17、ide APLENZIN Antidepressant; Antiobesity Agent Oral 905818-69-1 bupropion hydrochloride WELLBUTRIN Antidepressant Oral 04-Dec-1969 25-Jun-1991 31677-93-7 caffeine ALERT CNS Stimulant; Diuretic Oral;Other 26-Apr-1983 58-08-2 caffeine citrate CAFCIT CNS Stimulant Oral;Parent

18、eral;Other 69-22-7 caffeine sodium benzoate CAFFEINE SOD BENZ CNS Stimulant Parenteral calcium ACTICAL Oral;Other 7440-70-2 candesartan cilexetil ATACAND Antihypertensive; Angiotensin II Receptor Antagonist Oral 01-Jan-1919 18-Apr-2011 145040-37-5 capecitabine XELOD

19、A Antineoplastic Oral 17-Nov-1987 13-Jan-2011 154361-50-9 carvedilol COREG Antihypertensive; Adrenergic Blocker (Beta-) Oral 13-Apr-1978 05-Sep-2007 72956-09-3 carvedilol phosphate COREG CR Antihypertensive; Adrenergic Blocker (Beta-) Oral 610309-89-2 ceftriaxone sodium ROCEPH

20、IN Antibacterial (Antibiotic) Other;Parenteral 02-Apr-1977 14-Jul-1998 104376-79-6 celecoxib CELEBREX Anti-Inflammatory (Nonsteroidal); Cyclooxygenase-2 Inhibitor; Analgesic Oral 22-Sep-1992 30-Nov-2013 169590-42-5 cetuximab ERBITUX Antineoplastic Parenteral 08-Apr-1983 07-Jun-2015

21、 205923-56-4 chlorpheniramine maleate ANTAGONATE Antihistaminic Oral;Parenteral 04-Mar-1983 113-92-8 chlorpheniramine tannate PEDIATAN Antihistaminic Oral cholecalciferol VIT D Vitamin/Vitamin Source Oral 67-97-0 ciprofloxacin CIPRO Antibacterial (Synthetic) Parentera

22、l 03-Sep-1980 28-Oct-2003 85721-33-1 ciprofloxacin hydrochloride CIPRO Antibacterial (Synthetic) Ophthalmic;Otic;Oral 03-Sep-1980 28-Oct-2003 86393-32-0 ciprofloxacin lactate CIPRO IV Antibacterial (Synthetic) Parenteral 97867-33-9 citric acid Launched with generic name Oral;

23、Other 20-Oct-1998 77-92-9 clarithromycin BIAXIN Antibacterial (Antibiotic); Antiulcerative Oral 04-Jun-1980 23-May-2005 81103-11-9 clindamycin hydrochloride CLEOCIN Antibacterial (Antibiotic) Oral;Topical;Other 08-Feb-1965 17-Feb-1987 21462-39-5 clindamycin palmitate hydrochloride

24、 CLEOCIN Antibacterial (Antibiotic) Oral 25507-04-4 clindamycin phosphate CLEOCIN PHOSPHATE Antibacterial (Antibiotic) Parenteral;Vaginal;Topical 16-Dec-1966 30-Dec-1986 24729-96-2 clopidogrel bisulfate PLAVIX Antithrombotic Oral 13-Jul-1982 05-Jul-2003 120202-66-6 codeine pho

25、sphate CODEINE Analgesic (Narcotic); Antitussive Oral;Parenteral;Other 41444-62-6 codeine sulfate CODEINE SULF Analgesic (Narcotic); Antitussive Oral;Parenteral 6854-40-6 copper CU-7 Parenteral 27-Jan-2000 7440-50-8 cyanocobalamin BERUBIGEN Hematopoietic; Vitamin/Vitamin

26、 Source Nasal;Parenteral;Other;Oral 11-Feb-1983 68-19-9 cyclosporine SANDIMMUNE Immunosuppressant Ophthalmic;Parenteral;Other;Oral 07-Mar-1978 24-Jul-2004 59865-13-3 darbepoetin alfa ARANESP Hematopoietic Parenteral 13-Dec-1983 15-May-2024 209810-58-2 dexamethasone AEROSEB-DEX

27、Diagnostic Aid; Glucocorticoid; Antiallergic (Steroidal, Nasal); Antiasthmatic (Steroidal, Inhalant) Ophthalmic;Topical;Parenteral;Other;Oral 25-Nov-1960 02-Jun-2015 50-02-2 dexamethasone acetate DECADRON-LA Diagnostic Aid; Glucocorticoid; Antiallergic (Steroidal, Nasal); Antiasthmatic (Stero

28、idal, Inhalant) Other;Parenteral 55812-90-3 dexamethasone sodium phosphate DECADRON Diagnostic Aid; Glucocorticoid; Antiallergic (Steroidal, Nasal); Antiasthmatic (Steroidal, Inhalant) Nasal;Parenteral;Other;Ophthalmic 18-Apr-2008 2392-39-4 dextroamphetamine sulfate DEXAMPEX CNS Sti

29、mulant; Anorexic Oral 23-Aug-1999 51-63-8 dextromethorphan SCOT-TUSSIN DM Antitussive; Analgesic Oral 17-Jun-1991 125-71-3 dextromethorphan hydrobromide HOLD Antitussive; Analgesic Inhale;Topical;Other;Oral 17-Jun-1991 6700-34-1 dextromethorphan polistirex DELSYM Antitussive;

30、 Analgesic Oral dextromethorphan tannate AEROTUSS 12 Antitussive; Analgesic Oral dextrose GLUCOSE OPHTH Replenishers/Supplements; Antihypoglycemic Ophthalmic;Parenteral;Other;Oral 27-Aug-1996 50-99-7 dextrothyroxine sodium CHOLOXIN Antilipemic; Thyroid Hormone Oral 05-N

31、ov-1991 7054-08-2 diclofenac diethylamine VOLTAREN GEL Anti-Inflammatory (Nonsteroidal) Topical 78213-25-4 diclofenac epolamine FLECTOR Anti-Inflammatory (Nonsteroidal) Topical 119623-66-4 diclofenac potassium CATAFLAM Anti-Inflammatory (Nonsteroidal) Oral 15307-81-0 d

32、iclofenac sodium VOLTAREN Anti-Inflammatory (Nonsteroidal) Ophthalmic;Topical;Oral 08-Apr-1965 26-Jan-1988 15307-79-6 diltiazem hydrochloride CARDIZEM Antihypertensive; Vasodilator (Coronary); Antianginal; Calcium Channel Blocker Oral;Parenteral;Other 28-Oct-1967 09-Feb-1988 33286-22-5

33、 docetaxel anhydrous TAXOTERE Antineoplastic Parenteral 17-Jul-1986 14-May-2010 114977-28-5 doconexent DHA Oral 6217-54-5 donepezil hydrochloride ARICEPT Nootropic Oral 22-Jun-1987 31-Mar-2009 142057-77-0 duloxetine hydrochloride CYMBALTA Antidepressant; Serotonin Noradrena

34、line Reuptake Inhibitor (SNRI) Oral 22-Dec-1986 11-Sep-2007 136434-34-9 dutasteride AVODART Antiprostatic Hypertrophy; 5Alpha-Reductase Inhibitor Oral 17-Sep-1993 17-Sep-2013 164656-23-9 efavirenz SUSTIVA Antiviral; Reverse Transcriptase Inhibitor Oral 07-Aug-1992 07-Aug-2012 15459

35、8-52-4 emtricitabine EMTRIVA Antiviral Oral 01-Feb-1990 01-Feb-2010 143491-57-0 enalapril maleate VASOTEC Antihypertensive; Ace-Inhibitor Oral;Other 11-Dec-1978 18-Sep-2001 76095-16-4 enoxaparin sodium LOVENOX (PRESERVATIVE FREE) Antithrombotic Parenteral 679809-58-6 epoetin

36、alfa EPOGEN Hematopoietic Parenteral 29-Aug-2002 113427-24-0 ergocalciferol DELTALIN Vitamin/Vitamin Source Oral;Parenteral;Other 12-Oct-2000 50-14-6 erlotinib hydrochloride TARCEVA Antineoplastic Oral 30-Mar-1995 30-Mar-2015 183319-69-9 escitalopram oxalate LEXAPRO Antidepr

37、essant; Serotonin Uptake Inhibitor Oral 14-Jun-1988 08-Jun-2009 219861-08-2 esomeprazole magnesium NEXIUM Antiulcerative; Gastric Secretion Inhibitor Oral 04-Mar-1983 01-Mar-2008 217087-09-7 esomeprazole sodium NEXIUM IV Antiulcerative; Gastric Secretion Inhibitor Parenteral 04-Mar-1

38、983 01-Mar-2008 161796-78-7 estradiol ESTRACE Estrogen Oral;Vaginal;Transdermal;Topical;Parenteral;Other 16-Nov-1976 06-Mar-2007 50-28-2 estradiol (17beta-) ESTRASORB Estrogen Inhale;Transdermal estradiol acetate FEMRING Estrogen Oral;Other 4245-41-4 estradiol cypionate

39、 DEPO-ESTRADIOL Estrogen Oral;Parenteral;Other 313-06-4 estradiol valerate DELESTROGEN Estrogen Oral;Parenteral;Other 05-Aug-1983 979-32-8 estrogens conjugated PREMARIN Estrogen Oral;Vaginal;Parenteral etanercept ENBREL Cardiotonic; Antidiabetic; Analgesic (Non-narcotic);

40、 Immunosuppressant; Antiarthritic/Antirheumatic; Antipsoriatic; Anti-Inflammatory (Biological Response Modifier) Parenteral 25-Feb-1980 05-Sep-2009 185243-69-0 ethinyl estradiol ESTINYL Estrogen; Contraceptive (Oral) Oral 24-Jul-1975 28-Mar-1995 57-63-6 ezetimibe ZETIA Antilipemic Ora

41、l 09-Jul-1993 21-Mar-2014 163222-33-1 fenofibrate LIPIDIL Antilipemic Oral 31-Jan-1969 23-Sep-1992 49562-28-9 fentanyl DURAGESIC-100 Analgesic (Narcotic) Transdermal 21-Apr-1983 23-Jul-2004 437-38-7 fentanyl citrate SUBLIMAZE PRESERVATIVE FREE Analgesic (Narcotic) Oral;Parentera

42、l;Other 21-Apr-1983 23-Jul-2004 990-73-8 ferrous fumarate FEOSTAT Hematinic Oral 141-01-5 ferrous gluconate FERROUS GLUC Hematinic Oral 12389-15-0 ferrous sulfate FER-IN-SOL Hematinic Oral 7782-63-0 fexofenadine hydrochloride ALLEGRA Antihistaminic Oral 10-Apr-1979

43、 10-Apr-1999 138452-21-8 filgrastim NEUPOGEN(OLD) Hematopoietic; Antineutropenic Parenteral 04-Nov-1974 28-Mar-2005 121181-53-1 finasteride PROSCAR Antineoplastic; Antialopecia Agent; Antiprostatic Hypertrophy; 5Alpha-Reductase Inhibitor; Antifungal Oral 13-Apr-1978 13-Apr-1998 98319

44、26-7 fluticasone propionate CUTIVATE Glucocorticoid; Antiallergic (Steroidal, Nasal); Antiasthmatic (Steroidal, Inhalant); Anti-Inflammatory (Biological Response Modifier) Inhale;Topical;Nasal 15-Feb-1980 25-Mar-2003 80474-14-2 folic acid FOLICET Vitamin/Vitamin Source Oral;Parenteral;Ot

45、her 17-Oct-1995 59-30-3 formoterol fumarate FORADIL Bronchodilator; Adrenergic Agonist (Beta-); Antiasthmatic Inhale 05-Feb-1972 30-Nov-1993 43229-80-7 gabapentin NEURONTIN Antipsychotic; Analgesic (Non-narcotic); Antidepressant; Antimigraine; Anticonvulsant Oral;Other 21-Dec-1974 1

46、7-May-1994 60142-96-3 gemcitabine hydrochloride GEMZAR Antineoplastic Parenteral 10-Mar-1983 10-Mar-2003 122111-03-9 ginseng COLD FX Oral glatiramer acetate COPAXONE Immunomodulator; Neuroprotective Parenteral 21-Apr-1971 24-May-2014 147245-92-9 glimepiride AMARYL Antidi

47、abetic Oral 19-Dec-1979 06-Oct-2005 93479-97-1 glutamic acid hydrochloride (l-) GLUTAMIC ACID HCL Anxiolytic; Replenishers/Supplements; Acidifier Oral 138-15-8 glycine (l-) AMINOACETIC ACID 1.5% IN PLASTIC CONTAINER Antipruritic Other;Parenteral 56-40-6 guaifenesin MUCINEX E

48、xpectorant; Muscle Relaxant Oral 25-Feb-1981 93-14-1 hyaluronic acid RESTYLANE Antiarthritic/Antirheumatic Parenteral 07-Apr-1920 16-May-2008 9004-61-9 hydrochlorothiazide ESIDRIX Antihypertensive; Diuretic Oral 25-Sep-1964 29-Dec-1981 58-93-5 hydrocortisone ACTICORT Glucocorti

49、coid; Anti-Inflammatory (Biological Response Modifier) Oral;Topical;Rectal;Other 29-Mar-1978 50-23-7 hydrocortisone 17-butyrate LOCOID Glucocorticoid Topical 13609-67-1 hydrocortisone acetate CORTEF ACETATE Glucocorticoid Oral;Topical;Rectal;Parenteral;Other 50-03-3 hydrocort

50、isone cypionate CORTEF Glucocorticoid Oral 508-99-6 hydrocortisone sodium phosphate HYDROCORTONE Glucocorticoid Parenteral 6000-74-4 hydrocortisone sodium succinate A-HYDROCORT Glucocorticoid Parenteral 125-04-2 hydrocortisone valerate WESTCORT Glucocorticoid Topical

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